4 items found

Tags: opioid receptor affinity

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  • publication

    Effect of <i>N</i>-Alkyl and <i>N</i>-Alkenyl Substituents in Noroxymorphindo...

    The N-alkyl analogues (N-ethyl through N-heptyl), branched N-alkyl chain analogues (N-isopropyl, N-2-methylpropyl, and N-3-methylbutyl), and N-alkenyl analogues...
  • publication

    r37980778c78--a6e8c948fa454ae3cd105fb9c01cbb21

    Further modification of salvinorin A (1a), the major active component of Salvia divinorum, has resulted in the synthesis of novel neoclerodane diterpenes with opioid receptor...
  • publication

    r37980778c78--8a55b4d090be28a03d54dd1949a1eaaf

    Structural modification of salvinorin A, the active component of Salvia divinorum, has resulted in the synthesis of novel neoclerodane diterpenes with opioid receptor affinity...
  • publication

    Effects of the Substitution of Phe<sup>4</sup> in the Opioid Peptide [d-Ala<s...

    Phenylalanine at position 4 of the peptide dynorphin A (Dyn A) is an important residue for opioid receptor affinity and activity, but there is very little information available...