133 items found

Types: publication Groups: Open Access Tags: Cell Biology Chemical Sciences not elsewhere classified Evolutionary Biology Molecular Biology Pharmacology

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  • publication

    dedup_wf_001--4edd6b37544e4fc6acb3bb4fce0088b7

    A major bottleneck for the exploitation of data from the Kepler mission for stellar astrophysics and exoplanet research has been the lack of precise radii and evolutionary...
  • publication

    r37980778c78--45c77806280e278526960e808d2b7b2b

    Electrolysis of benzylthiocyanate, benzyl chloride, p-methylbenzyl chloride, p-methoxybenzyl chloride, or toluene in acetonitrile, at platinum electrodes in a two compartments...
  • publication

    Open Access Für Forschungsergebnisse. Forschungsdatenmanagement In Der Praxis

    Open Access für Forschungsergebnisse: Forschungsdatenmanagement in der Praxis Die Technische Universität Berlin unterstützt den offenen Zugang zu Forschungsdaten und...
  • publication

    Datenkuratierung In Den Sozial- Und Wirtschaftswissenschaften : Qualität Stat...

    Die Ziele der Open-Access-Bewegung sind klar umrissen: Alle Ergebnisse öffentlich finanzierter Forschung sollen der Gesellschaft zur Verfügung gestellt werden. Damit Wissen zum...
  • publication

    dedup_wf_001--2a5b8cddfaf4c65ddc0784cec145e2b8

    Im Moment herrscht unter den EthnologInnen noch Unklarheit über die Praxis von Archivierung und Nachnutzung von qualitativen Forschungsdaten. Zum einen gibt es ein solches...
  • publication

    Discovery of 1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9<i>H</i>-purin-6-yl]-4...

    We report the structure−activity relationships, design, and synthesis of the novel cannabinoid type 1 (CB1) receptor antagonist 3a (CP-945,598). Compound 3a showed subnanomolar...
  • publication

    r37980778c78--4816a1a6e4d6a60d570bdbb6d414ddf1

    In a previous study, we identified (−)-N-[(1R,4S,5S,7R)-5-(3-hydroxyphenyl)-4-methyl-2-(3-phenylpropyl)-2-azabicyclo[3.3.1]non-7-yl]-3-(1-piperidinyl)propanamide (5a, KAA-1) as...
  • publication

    r37980778c78--cd96dd5edfa917659346fa029ee432fc

    Spiro[1H-indene-1,4‘-piperidine] Derivatives As Potent and Selective Non-Peptide Human Somatostatin Receptor Subtype 2 (sst2) Agonists
  • publication

    Synthesis and Structure−Activity Relationship of Fluoro Analogues of 8-{2-[4-...

    We have discovered high-affinity antagonists (exemplified by 11 and 12) that are the most selective for α1d-adrenergic receptors (α1d-AR) reported to date. In cloned receptor...
  • publication

    Biohacking in Africa: A Tool for Justice, Empowerment, and Development

    SOHA project evidences on: obstacles to the adoption of Open Science in Haiti and Africa Panel on Inclusion and Diversity MIT-MediaLab 22 – 24 september 2017
  • publication

    dedup_wf_001--2b2407fcc86efdaecd554b355ffe5580

    Open-Access-Services der Technischen Universität Berlin Die Technische Universität Berlin hat mit der Unterzeichnung der "Berlin Declaration on Open Access to Knowledge in the...
  • publication

    Renormalization-Group Equations Of Neutrino Masses And Flavor Mixing Paramete...

    We apply the general idea of renormalization-group equations (RGEs) to understand how neutrino masses and flavor mixing parameters evolve when neutrinos propagate in a medium....
  • publication

    r37980778c78--98ad233a19199dd6829c44ca4f4531f4

    A functional cell-based screen identified 3-(4-chlorophenyl)-3-(2-(dimethylamino)ethyl)isochroman-1-one hydrochloride (AC-7954, 1) as a nonpeptidic agonist of the urotensin-II...
  • publication

    Synthesis and Structure−Activity Relationships of Cyanoguanidine-Type and Str...

    Recently, we identified high-affinity human histamine H3 (hH3R) and H4 receptor (hH4R) ligands among a series of NG-acylated imidazolylpropylguanidines, which were originally...
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    Open Access – Ein Vorschlag zur Klassifikation und Operationalisierung

    Der Begriff Open Access bezeichnet nicht nur eine bestimmte Art des wissenschaftlichen Publizierens – nämlich den leserseitig kostenlosen, freien Zugang zu Forschungsergebnissen...
  • publication

    Design, Synthesis, and SAR Study of a Series of <i>N</i>-Alkyl-<i>N</i><i>‘</...

    The prostanoid thromboxane (TX)A2 exerts its proaggregant and constrictive actions upon binding to the specific TXA2 receptor (TP), a member of the G-protein coupled receptor...
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    New 5-Hydroxytryptamine<sub>1A</sub> Receptor Ligands Containing a Norbornene...

    New arylpiperazine derivatives were prepared to identify highly selective and potent ligands for the 5-hydroxytryptamine 1A (5-HT1A) receptor as potential pharmacological tools...
  • publication

    Open Access : Von Inklusion Zu Exklusivität?

    Open Access scheint sich gewandelt zu haben. Um die Jahrtausendwende wurde er in Fach- und journalistischen Publikationen romantisierend dargestellt und war in ein...
  • publication

    5-(4-Chlorophenyl)-4-methyl-3-(1-(2- phenylethyl)piperidin-4-yl)isoxazole:  A...

    5-(4-Chlorophenyl)-4-methyl-3-(1-(2- phenylethyl)piperidin-4-yl)isoxazole:  A Potent, Selective Antagonist at Human Cloned Dopamine D4 Receptors
  • publication

    r37980778c78--e25f6b5df1b3d5c1f35b5060e3a6ddb9

    Following the discovery of the human histamine H4 receptor, a high throughput screen of our corporate compound collection identified compound 6 as a potential lead....