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Rationale, Design, and Synthesis of Novel Phenyl Imidazoles as Opioid Recepto...
A small series of novel, imidazoles 4 have been prepared that exhibit very good binding affinities for the δ and μ opioid receptors (ORs), as well as demonstrate potent agonist... -
Synthesis and Evaluation of a Full-Agonist Orvinol for PET-Imaging of Opioid ...
Antagonist radiotracers have shown only a low sensitivity for detecting competition from high-efficacy agonists at opioid receptors (ORs) in vivo. We report that [11C]PEO binds...
